A REACTION BETWEEN α-KETONIC ACIDS AND α-AMINO ACIDS
نویسندگان
چکیده
منابع مشابه
Coupling reaction between electron-rich pyrimidinones and α-amino acids promoted by phosphonium salts.
Coupling reaction between electron-rich 2-morpholino-4(3H)-pyrimidinone and nucleophilic side chains of several natural α-amino acids promoted by phosphonium salt has been developed to prepare new optically active pyrimidin-4-yl amino acids. The best results were obtained using a two-step method through the easily available benzotriazolyl-1-oxy intermediate. A detailed optimization study of thi...
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ژورنال
عنوان ژورنال: Journal of Biological Chemistry
سال: 1934
ISSN: 0021-9258
DOI: 10.1016/s0021-9258(18)75369-6